Synonym: trans-(1S,2S)-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]benzeneacetamide hydrochloride hydrate
Empirical Formula (Hill Notation): C19H26Cl2N2O HCl xH2O
Molecular Weight: 405.79 (anhydrous basis)
CAS Number: 114528-79-9 (anhydrous)
ssay
98% (HPLC) | |
form | solid |
optical activity | []22/D 36.05, c = 0.73 in methanol(lit.) |
storage condition | desiccated |
color | white |
solubility | H2O: soluble13 mg/mL |
storage temp. | 2-8C |
Gene Information | human ... OPRK1(4986) |
Potent opioid receptor agonist; more potent enantiomer of ()-trans-U-50488.
()-trans-(1S,2S)-U-50488 hydrochloride hydrate is soluble in water at 13 mg/ml.
()-trans-(1S,2S)-U-50488 hydrochloride hydrate (U-50488) has been used as a -opioid receptor (KOR) agonist has been used to study its effect on the increase of tidal volumes in adult red-eared slider turtles (Trachemys scripta)[1].