Synonym: (R)-N6-(1-Methyl-2-phenylethyl)adenosine, N6-(L-2-Phenylisopropyl)adenosine, R-()-PIA
Empirical Formula (Hill Notation): C19H23N5O4
Molecular Weight: 385.42
CAS Number: 38594-96-6
form
solid | |
potency | 1.17 nM Ki for A1 receptors (using [3H]CHA in rat forebrain preparations) |
color | white |
solubility | H2O: slightly soluble0.3 mg/mL (Solutions may be stored for several days at 4C.) |
45% (w/v) aq 2-hydroxypropyl--cyclode | |
storage temp. | 2-8C |
Gene Information | human ... ADORA1(134) |
25 mg in poly bottle
50, 100 mg in glass bottle
A1 adenosine receptor agonist. Affinity for adenosine receptor is approx. 100 that of the (+)-isomer.
This compound is also offered as part of Sigmas Library of Pharmacologically Active Compounds (LOPAC1280), a biologically annotated collection of high-quality, ready-to-screen compounds.
This compound is featured on the Adenosine Receptors page of the Handbook of Receptor Classification and Signal Transduction.